TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 7.70E+4nMAssay Description:Antagonist activity at rat alpha3beta4 nicotinic receptor expressed in KXalpha3beta4R2 cells assessed as nicotine-induced calcium fluorescenceMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 9.40E+4nMAssay Description:Antagonist activity at rat alpha3beta4 nicotinic receptor expressed in KXalpha3beta4R2 cells assessed as nicotine-induced calcium fluorescenceMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at rat alpha3beta4 nicotinic receptor expressed in KXalpha3beta4R2 cells assessed as nicotine-induced 86Rb+ effluxMore data for this Ligand-Target Pair